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4GHI

Crystal structure of the high affinity heterodimer of HIF2 alpha and ARNT C-terminal PAS domains in complex with a benzoxadiazole antagonist

Functional Information from PDB Data
site_idAC1
Number of Residues15
DetailsBINDING SITE FOR RESIDUE 0X3 A 401
ChainResidue
APHE244
ALEU296
ASER304
ATYR307
AILE337
ACYS339
AASN341
ASER246
AHIS248
AMET252
AALA277
ATYR281
AMET289
ASER292
AHIS293

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues43
DetailsDomain: {"description":"PAC"}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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