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4EQZ

Crystal structure of human DOT1L in complex with inhibitor FED2

Functional Information from GO Data
ChainGOidnamespacecontents
A0031151molecular_functionhistone H3K79 methyltransferase activity
A0051726biological_processregulation of cell cycle
Functional Information from PDB Data
site_idAC1
Number of Residues18
DetailsBINDING SITE FOR RESIDUE AW0 A 501
ChainResidue
APRO130
AGLY221
AASP222
APHE223
APHE239
AVAL240
AASN241
APHE245
ATYR312
AHOH645
APHE131
AASP161
AGLY163
ASER164
AGLY165
AVAL169
AGLU186
ALYS187

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues14
DetailsBinding site: {}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsModified residue: {"description":"Phosphoserine","evidences":[{"source":"PubMed","id":"23186163","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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