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4EBK

Crystal structure of aminoglycoside 4'-O-adenylyltransferase ANT(4')-IIb, tobramycin-bound

Functional Information from GO Data
ChainGOidnamespacecontents
A0016740molecular_functiontransferase activity
A0016779molecular_functionnucleotidyltransferase activity
B0016740molecular_functiontransferase activity
B0016779molecular_functionnucleotidyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues13
DetailsBINDING SITE FOR RESIDUE TOY A 301
ChainResidue
AGLU122
AHOH638
BASP40
BGLU51
BTYR53
AGLU124
AGLU126
AASP127
AGLU130
AHOH431
AHOH505
AHOH518
AHOH627

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 302
ChainResidue
ATYR28
AALA29
AARG98
AASP228
APRO229
AASP230

site_idAC3
Number of Residues1
DetailsBINDING SITE FOR RESIDUE IOD A 303
ChainResidue
BHIS3

site_idAC4
Number of Residues2
DetailsBINDING SITE FOR RESIDUE IOD A 306
ChainResidue
ASER150
ATHR153

site_idAC5
Number of Residues2
DetailsBINDING SITE FOR RESIDUE IOD A 307
ChainResidue
AARG7
AARG11

site_idAC6
Number of Residues2
DetailsBINDING SITE FOR RESIDUE IOD A 308
ChainResidue
ACYS198
AMSE217

site_idAC7
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CL A 309
ChainResidue
AGLU179
BHOH631

site_idAC8
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CL A 310
ChainResidue
AGLN152
ALYS156
ACL319
BGLN152

site_idAC9
Number of Residues1
DetailsBINDING SITE FOR RESIDUE CL A 311
ChainResidue
AHOH524

site_idBC1
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CL A 313
ChainResidue
AHOH426
AHOH633

site_idBC2
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CL A 314
ChainResidue
AGLN-1
AALA120

site_idBC3
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CL A 316
ChainResidue
AARG175
BLYS134

site_idBC4
Number of Residues3
DetailsBINDING SITE FOR RESIDUE CL A 317
ChainResidue
ALYS134
BARG30
BHOH621

site_idBC5
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CL A 318
ChainResidue
AHOH609
BLYS134

site_idBC6
Number of Residues3
DetailsBINDING SITE FOR RESIDUE CL A 319
ChainResidue
ALYS156
ACL310
BLYS156

site_idBC7
Number of Residues3
DetailsBINDING SITE FOR RESIDUE CL B 301
ChainResidue
ALYS134
AHOH612
BARG175

site_idBC8
Number of Residues16
DetailsBINDING SITE FOR RESIDUE TOY B 302
ChainResidue
AASP40
AGLU51
ATYR53
AHOH421
BGLU122
BGLU124
BGLU126
BASP127
BGLU130
BHOH414
BHOH489
BHOH496
BHOH510
BHOH560
BHOH616
BHOH626

site_idBC9
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO B 303
ChainResidue
AALA183
APRO185
BPRO185
BARG186

site_idCC1
Number of Residues2
DetailsBINDING SITE FOR RESIDUE IOD B 305
ChainResidue
BCYS198
BMSE217

site_idCC2
Number of Residues1
DetailsBINDING SITE FOR RESIDUE IOD B 307
ChainResidue
BGLU179

site_idCC3
Number of Residues2
DetailsBINDING SITE FOR RESIDUE IOD B 309
ChainResidue
BSER150
BTHR153

site_idCC4
Number of Residues3
DetailsBINDING SITE FOR RESIDUE CL B 310
ChainResidue
BMSE240
BHOH431
BHOH581

site_idCC5
Number of Residues1
DetailsBINDING SITE FOR RESIDUE CL B 311
ChainResidue
BHOH420

site_idCC6
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CL B 313
ChainResidue
BARG175
BGLU179

site_idCC7
Number of Residues1
DetailsBINDING SITE FOR RESIDUE CL B 314
ChainResidue
BGLY31

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PDB entries from 2024-07-24

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