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4D6Q

crystal structure of human JMJD2D in complex with 2,4-PDCA

Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 1341
ChainResidue
ACYS238
AHIS244
ACYS310
ACYS312

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE NI A 1342
ChainResidue
AHIS192
AGLU194
AHIS280
APD21343
AHOH2287

site_idAC3
Number of Residues13
DetailsBINDING SITE FOR RESIDUE PD2 A 1343
ChainResidue
ATYR136
APHE189
AHIS192
AGLU194
ALYS210
ALYS245
AHIS280
ANI1342
AEDO1348
AHOH2234
AHOH2286
AHOH2287
AHOH2293

site_idAC4
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 1344
ChainResidue
ALYS150
AGLN151
ATRP152
AASN153
AHIS156
AHOH2054
AHOH2055

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1345
ChainResidue
APRO251
ATHR252
ALYS255
AARG263
AHOH2405

site_idAC6
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1346
ChainResidue
APHE118
AGLU122
AARG263
AILE264
ATHR265
AHOH2406

site_idAC7
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 1347
ChainResidue
ALYS124
ALYS127
AASN128

site_idAC8
Number of Residues8
DetailsBINDING SITE FOR RESIDUE EDO A 1348
ChainResidue
ATYR179
ATYR181
AGLU194
AALA292
APD21343
AHOH2287
AHOH2293
AHOH2370

site_idAC9
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 1349
ChainResidue
AARG60
AGLU61
ATHR62
AHOH2120
AHOH2123
AHOH2264

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:B2RXH2
ChainResidueDetails
ATYR136
AASN202
ALYS210
ALYS245

site_idSWS_FT_FI2
Number of Residues3
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00538, ECO:0000305|PubMed:26741168
ChainResidueDetails
AHIS192
AGLU194
AHIS280

site_idSWS_FT_FI3
Number of Residues4
DetailsBINDING: BINDING => ECO:0007744|PDB:5F5A, ECO:0007744|PDB:5F5C
ChainResidueDetails
ACYS238
AHIS244
ACYS310
ACYS312

site_idSWS_FT_FI4
Number of Residues2
DetailsMOD_RES: PolyADP-ribosyl glutamic acid => ECO:0000269|PubMed:23102699
ChainResidueDetails
AGLU26
AGLU27

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PDB entries from 2024-05-01

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