Loading
PDBj
MenuPDBj@FacebookPDBj@X(formerly Twitter)PDBj@BlueSkyPDBj@YouTubewwPDB FoundationwwPDBDonate
RCSB PDBPDBeBMRBAdv. SearchSearch help

4CV9

MPS1 kinase with 3-aminopyridin-2-one inhibitors

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues12
DetailsBINDING SITE FOR RESIDUE W2K A 1795
ChainResidue
AILE531
ASER611
ALEU654
AILE663
AALA551
ALYS553
AMET602
AGLU603
ACYS604
AGLY605
AASN606
AASP608

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 1796
ChainResidue
ALYS521
AASP590
ATYR591
AGLU784

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1797
ChainResidue
AASP595
AHIS636
AHIS639
AILE782
AEDO1799
AHOH2027

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 1798
ChainResidue
AILE549
ATYR550
ATYR589
AHOH2006

site_idAC5
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 1799
ChainResidue
ATHR594
AASP595
AGLN596
APRO783
AEDO1797
AHOH2013
AHOH2030

site_idAC6
Number of Residues2
DetailsBINDING SITE FOR RESIDUE EDO A 1800
ChainResidue
AILE531
ASER533

site_idAC7
Number of Residues1
DetailsBINDING SITE FOR RESIDUE DMS A 1801
ChainResidue
ATYR599

Functional Information from PROSITE/UniProt
site_idPS00108
Number of Residues13
DetailsPROTEIN_KINASE_ST Serine/Threonine protein kinases active-site signature. IvHsDLKpaNFLI
ChainResidueDetails
AILE643-ILE655

site_idPS00107
Number of Residues23
DetailsPROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. IGSGGSSKVFqVlnekkqi...........YAIK
ChainResidueDetails
AILE531-LYS553

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsActive site: {"description":"Proton acceptor","evidences":[{"source":"PROSITE-ProRule","id":"PRU00159","evidenceCode":"ECO:0000255"},{"source":"PROSITE-ProRule","id":"PRU10027","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues9
DetailsBinding site: {"evidences":[{"source":"PROSITE-ProRule","id":"PRU00159","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

246905

PDB entries from 2025-12-31

PDB statisticsPDBj update infoContact PDBjnumon