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4CFK

N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH LY294002

Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE GOL A 1169
ChainResidue
ATRP81
AGLN85
AASP96
AHOH2145
AHOH2235
AHOH2236

site_idAC2
Number of Residues9
DetailsBINDING SITE FOR RESIDUE LY2 A 1170
ChainResidue
AVAL87
ALEU92
ALEU94
AASN140
AILE146
AHOH2148
ATRP81
APRO82
APHE83

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1171
ChainResidue
AILE100
AILE101
ALYS102
ATHR103
AASN135
AHOH2238

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

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PDB entries from 2024-06-12

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