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4C7H

Leismania major N-myristoyltransferase in complex with a peptidomimetic (-NH2) molecule

Functional Information from GO Data
ChainGOidnamespacecontents
A0004379molecular_functionglycylpeptide N-tetradecanoyltransferase activity
A0005829cellular_componentcytosol
A0006499biological_processN-terminal protein myristoylation
A0016740molecular_functiontransferase activity
A0016746molecular_functionacyltransferase activity
A0046872molecular_functionmetal ion binding
A0072657biological_processprotein localization to membrane
Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE MG A 1422
ChainResidue
ALEU175
AGLU177
ALYS178
AARG179
ALEU180
ACOA1424
AMYA1425

site_idAC2
Number of Residues22
DetailsBINDING SITE FOR RESIDUE EN5 A 1423
ChainResidue
AASP85
AASN167
ATHR203
ATYR217
AHIS219
APHE232
ATYR253
AALA394
AGLY395
AASP396
AGLY397
ALEU399
AMYA1425
ADMS1428
AHOH2179
AHOH2182
AHOH2300
AHOH2499
AHOH2518
AHOH2531
AASP83
AASP84

site_idAC3
Number of Residues29
DetailsBINDING SITE FOR RESIDUE COA A 1424
ChainResidue
AHIS12
AALA13
APHE14
ATRP15
AASN79
AVAL81
ALEU169
ACYS170
AVAL171
AARG176
AGLU177
ALYS178
AARG179
ALEU180
AALA181
APRO182
ATHR203
ALEU208
AMG1422
AENF1426
AHOH2003
AHOH2314
AHOH2532
AHOH2533
AHOH2534
AHOH2537
AHOH2538
AHOH2539
AHOH2540

site_idAC4
Number of Residues36
DetailsBINDING SITE FOR RESIDUE MYA A 1425
ChainResidue
AHIS12
AALA13
APHE14
ATRP15
AASN79
ATYR80
AVAL81
APHE168
ALEU169
ACYS170
AVAL171
AARG176
AGLU177
ALYS178
AARG179
ALEU180
AALA181
APRO182
ATHR189
AVAL192
ATRP198
ATYR202
ATHR203
ALEU208
ATYR404
AMG1422
AEN51423
AHOH2003
AHOH2314
AHOH2532
AHOH2533
AHOH2534
AHOH2537
AHOH2538
AHOH2539
AHOH2540

site_idAC5
Number of Residues26
DetailsBINDING SITE FOR RESIDUE ENF A 1426
ChainResidue
ALEU169
ATHR189
AVAL192
ATRP198
ATYR202
ATHR203
ATYR217
AHIS219
APHE232
AALA394
AGLY395
AASP396
AGLY397
ALEU399
ATYR404
ACOA1424
ADMS1428
AHOH2179
AHOH2182
AHOH2499
AHOH2518
ATYR80
AASP83
AASP84
AASP85
APHE168

site_idAC6
Number of Residues6
DetailsBINDING SITE FOR RESIDUE DMS A 1427
ChainResidue
APHE90
ATYR92
ATYR217
ATYR345
AHOH2473
AHOH2531

site_idAC7
Number of Residues6
DetailsBINDING SITE FOR RESIDUE DMS A 1428
ChainResidue
APHE88
APHE90
ASER330
AEN51423
AENF1426
AHOH2473

Functional Information from PROSITE/UniProt
site_idPS00975
Number of Residues9
DetailsNMT_1 Myristoyl-CoA:protein N-myristoyltransferase signature 1. EINFLCvHK
ChainResidueDetails
AGLU165-LYS173

site_idPS00976
Number of Residues7
DetailsNMT_2 Myristoyl-CoA:protein N-myristoyltransferase signature 2. KFGaGDG
ChainResidueDetails
ALYS391-GLY397

237992

PDB entries from 2025-06-25

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