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4BW1

The first bromodomain of human BRD4 in complex with 3,5 dimethylisoxaxole ligand

Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 1169
ChainResidue
ASER51
AASN52
ALYS55
ALYS57
ATRP81
AS5B1172
AHOH2027

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1170
ChainResidue
ALYS112
AHOH2174
AHOH2175
APRO86
AGLY108

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 1171
ChainResidue
AILE100
AILE101
ALYS102
ATHR103
AASN135
AHOH2114

site_idAC4
Number of Residues14
DetailsBINDING SITE FOR RESIDUE S5B A 1172
ChainResidue
ASER51
ALYS57
ATRP81
APRO82
APHE83
ALEU92
ALEU94
AASN116
AASN140
AEDO1169
AHOH2087
AHOH2091
AHOH2106
AHOH2177

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

223790

PDB entries from 2024-08-14

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