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4BJC

Crystal structure of human tankyrase 2 in complex with Rucaparib

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE RPB A 2162
ChainResidue
AHIS1031
AHOH2089
AGLY1032
ATYR1060
APHE1061
AALA1062
ALYS1067
ASER1068
ATYR1071
AGLU1138

site_idAC2
Number of Residues8
DetailsBINDING SITE FOR RESIDUE SO4 A 2163
ChainResidue
AARG977
AHIS979
AARG980
ALYS1067
AGLN1070
AASN1132
AHOH2028
AHOH2067

site_idAC3
Number of Residues8
DetailsBINDING SITE FOR RESIDUE SO4 A 2163
ChainResidue
AARG977
AHIS979
AARG980
ALYS1067
AGLN1070
AASN1132
AHOH2028
AHOH2067

site_idAC4
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 A 2164
ChainResidue
AASN990
AARG991
AMET1158
AARG1159
APRO1160
AGLU1161
AHOH2035

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 2165
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:O95271
ChainResidueDetails
ACYS1081
AHIS1084
ACYS1089
ACYS1092

223532

PDB entries from 2024-08-07

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