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4APU

PR X-Ray structures in agonist conformations reveal two different mechanisms for partial agonism in 11beta-substituted steroids

Functional Information from PDB Data
site_idAC1
Number of Residues13
DetailsBINDING SITE FOR RESIDUE OR8 A 1933
ChainResidue
ALEU715
APHE778
AMET801
ALEU887
ACYS891
ALEU718
AASN719
ALEU721
AGLY722
AGLN725
ATRP755
AMET756
AMET759

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 1934
ChainResidue
APRO737
AGLY738
AARG740
AASN741

site_idAC3
Number of Residues20
DetailsBINDING SITE FOR RESIDUE A2K B 1933
ChainResidue
BLEU718
BASN719
BLEU721
BGLY722
BGLN725
BTRP755
BMET756
BMET759
BARG766
BPHE778
BLEU797
BMET801
BTYR890
BCYS891
BTHR894
BPHE905
BMET909
BILE913
BHOH2018
BHOH2030

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"9620806","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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