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4ALH

N-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 3,5 dimethyl-4-phenyl-1,2- oxazole

Replaces:  4A9P
Functional Information from PDB Data
site_idAC1
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 1183
ChainResidue
AGLN94
AHOH2130
BTRP97

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1184
ChainResidue
ATRP97
AA9P1185
AHOH2114
AHOH2132
BGLN94

site_idAC3
Number of Residues7
DetailsBINDING SITE FOR RESIDUE A9P A 1185
ChainResidue
APHE99
ALEU108
ALEU110
AASN156
AEDO1184
AHOH2066
APRO98

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE A9P B 1184
ChainResidue
BPRO98
BPHE99
BASN156
BHOH2033

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE A9P C 1183
ChainResidue
CPRO98
CLEU108
CLEU110
CASN156
CHOH2028

site_idAC6
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 C 1184
ChainResidue
BARG100
BHOH2010
CARG128
CASN132
CTYR134
CHOH2043
CHOH2073

site_idAC7
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 1186
ChainResidue
AARG100
AHOH2025
AHOH2027

site_idAC8
Number of Residues1
DetailsBINDING SITE FOR RESIDUE SO4 A 1187
ChainResidue
AARG129

site_idAC9
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 B 1185
ChainResidue
AGLN167
ALYS171
ALEU174
BGLN143
BASN146
BTHR147
BHOH2096

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFrqpvDavklglpDYHkiIkqpMdmgtIkrrlenny..Ywaasecmqdfnt.MftNCyiY
ChainResidueDetails
AALA96-TYR155

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues12
DetailsBINDING: BINDING => ECO:0000269|PubMed:37731000, ECO:0007744|PDB:8SB6
ChainResidueDetails
AASP112
ATYR155
AASN156
ALYS157
BASP112
BTYR155
BASN156
BLYS157
CASP112
CTYR155
CASN156
CLYS157

site_idSWS_FT_FI2
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:20048151, ECO:0007744|PDB:2DVQ, ECO:0007744|PDB:2DVS
ChainResidueDetails
AASP160
AASP161
BASP160
BASP161
CASP160
CASP161

219869

PDB entries from 2024-05-15

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