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4A9O

N-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 5 ethyl-3-methyl-4-phenyl-1, 2-oxazole

Functional Information from PDB Data
site_idAC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1189
ChainResidue
AGLN94
AHOH2032
AHOH2176
AHOH2177
BTRP97

site_idAC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE A9O A 1190
ChainResidue
AASN156
AHOH2082
BEDO1184
APRO98
APHE99
ALEU110
ATYR155

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 1191
ChainResidue
AARG100
AHOH2024
AHOH2027
AHOH2029

site_idAC4
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 1192
ChainResidue
AARG128
AARG129
AHOH2115

site_idAC5
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO B 1184
ChainResidue
ATRP97
AA9O1190
BGLN94
BHOH2019
BHOH2129
BHOH2130

site_idAC6
Number of Residues6
DetailsBINDING SITE FOR RESIDUE A9O B 1185
ChainResidue
BPRO98
BPHE99
BLEU110
BTYR155
BASN156
BHOH2045

site_idAC7
Number of Residues5
DetailsBINDING SITE FOR RESIDUE A9O C 1183
ChainResidue
CPRO98
CLEU110
CTYR155
CASN156
CHOH2036

site_idAC8
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 C 1184
ChainResidue
BARG100
CARG128
CASN132
CTYR134
CHOH2060
CHOH2099
CHOH2100

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFrqpvDavklglpDYHkiIkqpMdmgtIkrrlenny..Ywaasecmqdfnt.MftNCyiY
ChainResidueDetails
AALA96-TYR155

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues12
DetailsBINDING: BINDING => ECO:0000269|PubMed:37731000, ECO:0007744|PDB:8SB6
ChainResidueDetails
AASP112
CTYR155
CASN156
CLYS157
ATYR155
AASN156
ALYS157
BASP112
BTYR155
BASN156
BLYS157
CASP112

site_idSWS_FT_FI2
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:20048151, ECO:0007744|PDB:2DVQ, ECO:0007744|PDB:2DVS
ChainResidueDetails
AASP160
AASP161
BASP160
BASP161
CASP160
CASP161

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PDB entries from 2024-07-17

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