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4A9E

N-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 3-methyl-1,2,3,4- tetrahydroquinazolin-2-one

Functional Information from PDB Data
site_idAC1
Number of Residues6
DetailsBINDING SITE FOR RESIDUE 3PF A 1000
ChainResidue
APRO98
AVAL103
ALEU108
AASN156
AEDO1187
AHOH2060

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE 3PF B 1000
ChainResidue
BHOH2043
BVAL103
BLEU108
BASN156

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE 3PF C 1000
ChainResidue
CVAL103
CASN156
CILE162
CHOH2030

site_idAC4
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO B 1186
ChainResidue
AGLN94
BTRP97
BHOH2099

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE EDO A 1187
ChainResidue
ATRP97
A3PF1000
AHOH2134
BGLN94

site_idAC6
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 1188
ChainResidue
AVAL75
ALEU79
AGLN80
AHIS83
ALEU130
AASN133
AHOH2097

site_idAC7
Number of Residues2
DetailsBINDING SITE FOR RESIDUE EDO B 1187
ChainResidue
BARG128
BARG129

site_idAC8
Number of Residues8
DetailsBINDING SITE FOR RESIDUE SO4 C 1184
ChainResidue
BARG100
CARG128
CASN132
CTYR134
CHOH2044
CHOH2051
CHOH2074
CHOH2075

site_idAC9
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 1190
ChainResidue
ATRP97
AARG100
AHOH2018
AHOH2022

site_idBC1
Number of Residues2
DetailsBINDING SITE FOR RESIDUE SO4 A 1191
ChainResidue
AARG128
AARG129

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFrqpvDavklglpDYHkiIkqpMdmgtIkrrlenny..Ywaasecmqdfnt.MftNCyiY
ChainResidueDetails
AALA96-TYR155

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues12
DetailsBINDING: BINDING => ECO:0000269|PubMed:37731000, ECO:0007744|PDB:8SB6
ChainResidueDetails
AASP112
CTYR155
CASN156
CLYS157
ATYR155
AASN156
ALYS157
BASP112
BTYR155
BASN156
BLYS157
CASP112

site_idSWS_FT_FI2
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:20048151, ECO:0007744|PDB:2DVQ, ECO:0007744|PDB:2DVS
ChainResidueDetails
AASP160
AASP161
BASP160
BASP161
CASP160
CASP161

237992

PDB entries from 2025-06-25

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