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3ZRB

Structural basis for agonism and antagonism for a set of chemically related progesterone receptor modulators

Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE OR8 A 1000
ChainResidue
ALEU715
ATHR894
ALEU718
AASN719
ALEU721
AGLN725
AMET756
AMET759
AMET801
ACYS891

site_idAC2
Number of Residues11
DetailsBINDING SITE FOR RESIDUE ORC B 1000
ChainResidue
BLEU715
BLEU718
BASN719
BTRP755
BMET756
BMET759
BMET801
BTYR890
BCYS891
BPHE905
BMET909

site_idAC3
Number of Residues9
DetailsBINDING SITE FOR RESIDUE SO4 A 1933
ChainResidue
APRO737
AGLY738
AARG740
AASN741
AHOH2138
BPRO737
BGLY738
BARG740
BASN741

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL A 1934
ChainResidue
APRO737
AGLY738
AMET844
ASER847
AGOL1936

site_idAC5
Number of Residues7
DetailsBINDING SITE FOR RESIDUE GOL A 1935
ChainResidue
ATYR753
ATHR829
AHIS881
AHIS888
AILE920
AHOH2050
AHOH2114

site_idAC6
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL A 1936
ChainResidue
AGOL1934
AHOH2138
BLEU687
BGLY738
BSER847

site_idAC7
Number of Residues3
DetailsBINDING SITE FOR RESIDUE GOL B 1933
ChainResidue
BTYR890
BASN893
BTHR894

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"9620806","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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