Loading
PDBj
MenuPDBj@FacebookPDBj@X(formerly Twitter)PDBj@BlueSkyPDBj@YouTubewwPDB FoundationwwPDBDonate
RCSB PDBPDBeBMRBAdv. SearchSearch help

3ZR7

Structural basis for agonism and antagonism for a set of chemically related progesterone receptor modulators

Functional Information from PDB Data
site_idAC1
Number of Residues15
DetailsBINDING SITE FOR RESIDUE OR8 A 1000
ChainResidue
ALEU715
AMET801
ACYS891
ATHR894
APHE905
AMET909
AHOH2038
ALEU718
AASN719
AGLN725
ATRP755
AMET756
AMET759
ALEU763
APHE778

site_idAC2
Number of Residues14
DetailsBINDING SITE FOR RESIDUE OR8 B 1000
ChainResidue
BLEU715
BLEU718
BASN719
BGLN725
BTRP755
BMET756
BMET759
BPHE778
BMET801
BTYR890
BCYS891
BTHR894
BPHE905
BMET909

site_idAC3
Number of Residues3
DetailsBINDING SITE FOR RESIDUE GOL A 1933
ChainResidue
ATYR890
AASN893
ATHR894

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1934
ChainResidue
APRO737
AGLY738
AARG740
AASN741
AHOH2172

site_idAC5
Number of Residues8
DetailsBINDING SITE FOR RESIDUE GOL B 1933
ChainResidue
BTYR753
BTHR829
BHIS881
BHIS888
BILE920
BHOH2064
BHOH2142
BHOH2173

site_idAC6
Number of Residues6
DetailsBINDING SITE FOR RESIDUE GOL A 1935
ChainResidue
ALEU687
AGLY738
ASER847
AHOH2116
AHOH2120
AHOH2172

site_idAC7
Number of Residues7
DetailsBINDING SITE FOR RESIDUE GOL A 1936
ChainResidue
AGLU695
AGLN725
AARG766
ALYS822
AHOH2011
AHOH2173
AHOH2174

site_idAC8
Number of Residues7
DetailsBINDING SITE FOR RESIDUE GOL A 1937
ChainResidue
ATYR753
ATHR829
AHIS881
AHIS888
AILE920
AHOH2074
AHOH2136

site_idAC9
Number of Residues3
DetailsBINDING SITE FOR RESIDUE GOL A 1938
ChainResidue
AGLN752
AGLU911
AVAL912

site_idBC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE GOL B 1934
ChainResidue
BLEU687
BGLY738
BSER847
BHOH2050

site_idBC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE GOL B 1935
ChainResidue
BTYR890
BASN893
BTHR894
BGLN897
BHOH2147
BHOH2174

site_idBC3
Number of Residues8
DetailsBINDING SITE FOR RESIDUE GOL B 1936
ChainResidue
BGLU695
BPRO696
BGLN725
BARG766
BLYS822
BHOH2013
BHOH2175
BHOH2176

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"9620806","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

238895

PDB entries from 2025-07-16

PDB statisticsPDBj update infoContact PDBjnumon