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3W0P

Crystal structure of a thermostable mutant of aminoglycoside phosphotransferase APH(4)-Ia (D198A), ternary complex with ADP and hygromycin B

Functional Information from GO Data
ChainGOidnamespacecontents
A0005524molecular_functionATP binding
A0016301molecular_functionkinase activity
A0016310biological_processphosphorylation
A0046677biological_processresponse to antibiotic
Functional Information from PDB Data
site_idAC1
Number of Residues24
DetailsBINDING SITE FOR RESIDUE ADP A 401
ChainResidue
ALEU28
ALEU205
AILE215
AHOH506
AHOH530
AHOH532
AHOH538
AHOH540
AHOH560
AHOH579
AHOH589
ASER29
AHOH591
AHOH594
AHOH607
AHOH654
AHOH671
AALA36
AVAL47
APRO75
AARG93
AARG94
AALA95
ATHR99

site_idAC2
Number of Residues16
DetailsBINDING SITE FOR RESIDUE HY0 A 402
ChainResidue
AGLN101
AASP126
AALA198
ASER201
AASN202
AASN231
ATRP235
ATRP238
ALEU239
AGLN273
AASP285
AHOH588
AHOH601
AHOH625
AHOH664
AHOH732

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsACT_SITE: Proton acceptor => ECO:0000250
ChainResidueDetails
AALA198

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PDB entries from 2024-09-04

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