Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

3W0L

The crystal structure of Xenopus Glucokinase and Glucokinase Regulatory Protein complex

Functional Information from GO Data
ChainGOidnamespacecontents
A0001678biological_processintracellular glucose homeostasis
A0004340molecular_functionglucokinase activity
A0004396molecular_functionhexokinase activity
A0005524molecular_functionATP binding
A0005536molecular_functionD-glucose binding
A0005739cellular_componentmitochondrion
A0005829cellular_componentcytosol
A0005975biological_processcarbohydrate metabolic process
A0006006biological_processglucose metabolic process
A0006007biological_processglucose catabolic process
A0006096biological_processglycolytic process
A0008865molecular_functionfructokinase activity
A0016301molecular_functionkinase activity
A0016310biological_processphosphorylation
A0016773molecular_functionphosphotransferase activity, alcohol group as acceptor
A0019158molecular_functionmannokinase activity
A0019318biological_processhexose metabolic process
A0032024biological_processpositive regulation of insulin secretion
A0042593biological_processglucose homeostasis
A0045721biological_processnegative regulation of gluconeogenesis
A0045725biological_processpositive regulation of glycogen biosynthetic process
A0046835biological_processcarbohydrate phosphorylation
A0050796biological_processregulation of insulin secretion
A0051156biological_processglucose 6-phosphate metabolic process
B0004857molecular_functionenzyme inhibitor activity
B0005634cellular_componentnucleus
B0005654cellular_componentnucleoplasm
B0005737cellular_componentcytoplasm
B0005739cellular_componentmitochondrion
B0005829cellular_componentcytosol
B0009750biological_processresponse to fructose
B0019899molecular_functionenzyme binding
B0030246molecular_functioncarbohydrate binding
B0033132biological_processnegative regulation of glucokinase activity
B0042593biological_processglucose homeostasis
B0070095molecular_functionfructose-6-phosphate binding
B0097367molecular_functioncarbohydrate derivative binding
B1901135biological_processcarbohydrate derivative metabolic process
C0001678biological_processintracellular glucose homeostasis
C0004340molecular_functionglucokinase activity
C0004396molecular_functionhexokinase activity
C0005524molecular_functionATP binding
C0005536molecular_functionD-glucose binding
C0005739cellular_componentmitochondrion
C0005829cellular_componentcytosol
C0005975biological_processcarbohydrate metabolic process
C0006006biological_processglucose metabolic process
C0006007biological_processglucose catabolic process
C0006096biological_processglycolytic process
C0008865molecular_functionfructokinase activity
C0016301molecular_functionkinase activity
C0016310biological_processphosphorylation
C0016773molecular_functionphosphotransferase activity, alcohol group as acceptor
C0019158molecular_functionmannokinase activity
C0019318biological_processhexose metabolic process
C0032024biological_processpositive regulation of insulin secretion
C0042593biological_processglucose homeostasis
C0045721biological_processnegative regulation of gluconeogenesis
C0045725biological_processpositive regulation of glycogen biosynthetic process
C0046835biological_processcarbohydrate phosphorylation
C0050796biological_processregulation of insulin secretion
C0051156biological_processglucose 6-phosphate metabolic process
D0004857molecular_functionenzyme inhibitor activity
D0005634cellular_componentnucleus
D0005654cellular_componentnucleoplasm
D0005737cellular_componentcytoplasm
D0005739cellular_componentmitochondrion
D0005829cellular_componentcytosol
D0009750biological_processresponse to fructose
D0019899molecular_functionenzyme binding
D0030246molecular_functioncarbohydrate binding
D0033132biological_processnegative regulation of glucokinase activity
D0042593biological_processglucose homeostasis
D0070095molecular_functionfructose-6-phosphate binding
D0097367molecular_functioncarbohydrate derivative binding
D1901135biological_processcarbohydrate derivative metabolic process
Functional Information from PDB Data
site_idAC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 501
ChainResidue
AGLY220
ATHR221
AGLY403
ASER404
AARG440

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE NA A 502
ChainResidue
AMET231
AVAL234
AVAL237
AGLY239

site_idAC3
Number of Residues13
DetailsBINDING SITE FOR RESIDUE F6R B 701
ChainResidue
BCYS107
BGLY108
BTHR109
BSER110
BGLU153
BSER179
BCYS180
BSER183
BSER258
BARG259
BGLU347
BLYS513
BHOH811

site_idAC4
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 B 702
ChainResidue
BLEU80
BLYS81
BGLY84
BVAL286
BTHR287
BGLU288
BLEU291

site_idAC5
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 B 703
ChainResidue
BARG89
BVAL93
BLEU202

site_idAC6
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 C 501
ChainResidue
CGLY220
CTHR221
CSER404
CARG440

site_idAC7
Number of Residues5
DetailsBINDING SITE FOR RESIDUE NA C 502
ChainResidue
CMET231
CVAL234
CVAL237
CGLY239
CHOH604

site_idAC8
Number of Residues12
DetailsBINDING SITE FOR RESIDUE F6R D 701
ChainResidue
DCYS107
DGLY108
DTHR109
DGLU153
DSER179
DCYS180
DGLY181
DSER183
DSER258
DARG259
DGLU347
DLYS513

Functional Information from PROSITE/UniProt
site_idPS00378
Number of Residues26
DetailsHEXOKINASE_1 Hexokinase domain signature. LGFTFSFPvrhedIDkgiLlnWTKgF
ChainResidueDetails
ALEU139-PHE164

site_idPS01272
Number of Residues18
DetailsGCKR Glucokinase regulatory protein family signature. GPEgVSGSSRMKGGSatK
ChainResidueDetails
BGLY250-LYS267

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:23733961, ECO:0007744|PDB:3W0L
ChainResidueDetails
BCYS107
BGLU347
BLYS513
DCYS107
DGLU347
DLYS513

site_idSWS_FT_FI2
Number of Residues6
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:Q14397
ChainResidueDetails
BTHR109
BGLU153
BSER179
DTHR109
DGLU153
DSER179

223790

PDB entries from 2024-08-14

PDB statisticsPDBj update infoContact PDBjnumon