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3VHV

Mineralocorticoid receptor ligand-binding domain with non-steroidal antagonist

Functional Information from PDB Data
site_idAC1
Number of Residues16
DetailsBINDING SITE FOR RESIDUE LD1 A 1
ChainResidue
AHOH9
AMET845
AMET852
APHE941
ACYS942
ATHR945
AVAL954
APHE956
ALEU769
AASN770
ALEU772
AGLN776
AMET807
ALEU810
ASER811
APHE829

site_idAC2
Number of Residues16
DetailsBINDING SITE FOR RESIDUE LD2 A 2
ChainResidue
AHOH153
ALEU766
AALA844
AMET845
ATYR846
AGLU847
ALEU848
AILE900
ALYS901
AARG904
ATRP918
APHE941
ATYR944
ATHR945
ALEU952
AEDO985

site_idAC3
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 985
ChainResidue
ALD22
AHOH35
AHOH41
AARG896
ATHR897
AILE900
AGLU948

site_idAC4
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 986
ChainResidue
APRO788
ATYR899
AGLU902

site_idAC5
Number of Residues6
DetailsBINDING SITE FOR RESIDUE K A 3
ChainResidue
AHOH18
AHOH52
AHOH260
ATYR980
AARG983
ALYS984

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:15908963, ECO:0000269|PubMed:15967794, ECO:0007744|PDB:1YA3, ECO:0007744|PDB:2AA5, ECO:0007744|PDB:2AA6
ChainResidueDetails
AASN770
AGLN776
AARG817

site_idSWS_FT_FI2
Number of Residues1
DetailsBINDING: BINDING => ECO:0000269|PubMed:15967794, ECO:0007744|PDB:2AA5, ECO:0007744|PDB:2AA6
ChainResidueDetails
ATHR945

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PDB entries from 2024-07-24

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