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3UW5

Crystal structure of the BIR domain of MLIAP bound to GDC0152

Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 1001
ChainResidue
ACYS124
ACYS127
AHIS144
ACYS151

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 205
ChainResidue
AARG123
AHOH210
BARG136
BHOH196

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN B 1001
ChainResidue
BCYS127
BHIS144
BCYS151
BCYS124

site_idAC4
Number of Residues8
DetailsBINDING SITE FOR RESIDUE SO4 B 206
ChainResidue
BGLY117
BHIS118
BGLN119
BLYS121
BHOH175
BHOH180
BHOH201
BHOH203

site_idAC5
Number of Residues16
DetailsBINDING SITE FOR CHAIN Y OF GDC-0152
ChainResidue
AGLU106
ALEU107
BLYS121
BVAL122
BARG123
BGLY130
BLEU131
BGLN132
BSER133
BTRP134
BASP138
BGLU143
BTRP147
BHOH202
YHOH123
YHOH139

site_idAC6
Number of Residues12
DetailsBINDING SITE FOR CHAIN Z OF GDC-0152
ChainResidue
AVAL122
AARG123
AGLY130
ALEU131
AGLN132
ASER133
ATRP134
AASP138
AGLU143
ATRP147
BARG136
ZHOH160

Functional Information from PROSITE/UniProt
site_idPS01282
Number of Residues68
DetailsBIR_REPEAT_1 BIR repeat. EelRlasfyd.Wpltaevppellaa.AGFfHtghqDkvrCffCygglqsWkrgddpwteHakwfPgCqfL
ChainResidueDetails
AGLU87-LEU154

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues30
DetailsRegion: {"description":"Required for interaction with SEPTIN4 isoform ARTS","evidences":[{"source":"PubMed","id":"21695558","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues8
DetailsBinding site: {}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues6
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)","evidences":[{"source":"PubMed","id":"12747801","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues130
DetailsRepeat: {"description":"BIR"}
ChainResidueDetails

239492

PDB entries from 2025-07-30

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