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3U5J

Crystal Structure of the first bromodomain of human BRD4 in complex with Alprazolam

Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE 08H A 1
ChainResidue
ATRP81
AHOH226
APRO82
APHE83
ALEU92
AASP96
ALYS99
AASN140
AILE146
AHOH170

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 169
ChainResidue
AILE100
AILE101
ALYS102
ATHR103
AASN135
AHOH173

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 2
ChainResidue
APRO53
ALYS55
ALYS99
AHOH217
AHOH232
AHOH278

site_idAC4
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 3
ChainResidue
AARG58
ALEU63
ALEU114
AASN117
AHOH180
AHOH230
AHOH304

site_idAC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 4
ChainResidue
AARG68
AGLY143
AVAL147
AGLU151
AHOH218

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

223790

PDB entries from 2024-08-14

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