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3SX0

Crystal structure of Dot1l in complex with a brominated SAH analog

Functional Information from GO Data
ChainGOidnamespacecontents
A0031151molecular_functionhistone H3K79 methyltransferase activity
A0051726biological_processregulation of cell cycle
Functional Information from PDB Data
site_idAC1
Number of Residues18
DetailsBINDING SITE FOR RESIDUE SX0 A 421
ChainResidue
APRO133
ALYS187
AGLY221
AASP222
APHE223
APHE239
AASN241
APHE245
AHOH443
AHOH459
AGLY137
AGLU138
ATHR139
AASP161
AGLY163
ASER164
AGLN168
AGLU186

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 422
ChainResidue
AARG203
ALYS207
AHIS213
AHOH470

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues14
DetailsBinding site: {}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsModified residue: {"description":"Phosphoserine","evidences":[{"source":"PubMed","id":"23186163","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

248335

PDB entries from 2026-01-28

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