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3SPK

Tipranavir in Complex with a Human Immunodeficiency Virus Type 1 Protease Variant

Functional Information from GO Data
ChainGOidnamespacecontents
A0004190molecular_functionaspartic-type endopeptidase activity
A0006508biological_processproteolysis
B0004190molecular_functionaspartic-type endopeptidase activity
B0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues22
DetailsBINDING SITE FOR RESIDUE TPV A 100
ChainResidue
AARG8
AILE50
APRO81
ATHR82
AHOH208
AHOH232
AHOH340
BARG8
BLEU23
BASN25
BGLY48
AASN25
BGLY49
BILE50
BTHR82
AGLY27
AALA28
AASP29
AASP30
AILE47
AGLY48
AGLY49

site_idAC2
Number of Residues22
DetailsBINDING SITE FOR RESIDUE TPV B 100
ChainResidue
AARG8
ALEU23
AASN25
AALA28
AGLY49
AILE50
ATHR82
BARG8
BASN25
BGLY27
BALA28
BASP29
BASP30
BILE47
BGLY48
BGLY49
BILE50
BPRO81
BTHR82
BHOH107
BHOH154
BHOH338

219869

PDB entries from 2024-05-15

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