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3ROM

Crystal structure of human CD38 in complex with compound CZ-48

Functional Information from GO Data
ChainGOidnamespacecontents
A0061809molecular_functionNAD+ nucleotidase, cyclic ADP-ribose generating
B0061809molecular_functionNAD+ nucleotidase, cyclic ADP-ribose generating
Functional Information from PDB Data
site_idAC1
Number of Residues8
DetailsBINDING SITE FOR RESIDUE 48Z A 301
ChainResidue
ATRP125
ASER126
AARG127
ASER193
ASER220
ATHR221
APHE222
AGLU226

site_idAC2
Number of Residues10
DetailsBINDING SITE FOR RESIDUE 48Z B 301
ChainResidue
BSER126
BARG127
BGLU146
BSER193
BSER220
BTHR221
BPHE222
BGLU226
BHOH381
BTRP125

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsACT_SITE: ACT_SITE => ECO:0000305|PubMed:7961800
ChainResidueDetails
ACYS119
ACYS201
BCYS119
BCYS201

site_idSWS_FT_FI2
Number of Residues4
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:19159218
ChainResidueDetails
AASP100
AASP209
BASP100
BASP209

site_idSWS_FT_FI3
Number of Residues2
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255
ChainResidueDetails
AASP164
BASP164

site_idSWS_FT_FI4
Number of Residues2
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000269|PubMed:19159218, ECO:0000269|PubMed:19349973
ChainResidueDetails
AASP219
BASP219

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PDB entries from 2024-09-11

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