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3R8A

X-ray crystal structure of the nuclear hormone receptor PPAR-gamma in a complex with a compound with dual PPAR gamma agonism and Angiotensin II Type I receptor antagonism activity

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues15
DetailsBINDING SITE FOR RESIDUE HIG A 1
ChainResidue
AHOH154
AVAL339
ALEU340
AILE341
ASER342
AMET348
AMET364
AILE281
AGLY284
ACYS285
AARG288
ASER289
AILE326
ALEU330
ALEU333

site_idAC2
Number of Residues11
DetailsBINDING SITE FOR RESIDUE HIG B 1
ChainResidue
BHOH103
BGLY284
BCYS285
BARG288
BSER289
BILE326
BLEU340
BILE341
BSER342
BMET348
BMET364

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBINDING: BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
ChainResidueDetails
AGLN286
AHIS323
AHIS449
ATYR473
BGLN286
BHIS323
BHIS449
BTYR473

217705

PDB entries from 2024-03-27

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