3QZR
Human enterovirus 71 3C protease mutant E71A in complex with rupintrivir
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0004197 | molecular_function | cysteine-type endopeptidase activity |
A | 0005737 | cellular_component | cytoplasm |
A | 0006508 | biological_process | proteolysis |
A | 0008234 | molecular_function | cysteine-type peptidase activity |
A | 0019062 | biological_process | virion attachment to host cell |
A | 0030430 | cellular_component | host cell cytoplasm |
A | 0039618 | cellular_component | T=pseudo3 icosahedral viral capsid |
A | 0046718 | biological_process | symbiont entry into host cell |
B | 0004197 | molecular_function | cysteine-type endopeptidase activity |
B | 0005737 | cellular_component | cytoplasm |
B | 0006508 | biological_process | proteolysis |
B | 0008234 | molecular_function | cysteine-type peptidase activity |
B | 0019062 | biological_process | virion attachment to host cell |
B | 0030430 | cellular_component | host cell cytoplasm |
B | 0039618 | cellular_component | T=pseudo3 icosahedral viral capsid |
B | 0046718 | biological_process | symbiont entry into host cell |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 21 |
Details | BINDING SITE FOR RESIDUE AG7 A 501 |
Chain | Residue |
A | ARG39 |
A | ALA144 |
A | GLY145 |
A | CYS147 |
A | HIS161 |
A | ILE162 |
A | GLY163 |
A | GLY164 |
A | ASN165 |
A | PHE170 |
A | EDO184 |
A | HIS40 |
A | HOH252 |
A | HOH358 |
A | LEU125 |
A | ASN126 |
A | LEU127 |
A | SER128 |
A | LYS130 |
A | THR142 |
A | LYS143 |
site_id | AC2 |
Number of Residues | 7 |
Details | BINDING SITE FOR RESIDUE EDO A 184 |
Chain | Residue |
A | GLN22 |
A | GLY23 |
A | HIS24 |
A | HOH200 |
A | HOH260 |
A | HOH281 |
A | AG7501 |
site_id | AC3 |
Number of Residues | 21 |
Details | BINDING SITE FOR RESIDUE AG7 B 501 |
Chain | Residue |
B | ARG39 |
B | HIS40 |
B | LEU125 |
B | ASN126 |
B | LEU127 |
B | SER128 |
B | LYS130 |
B | THR142 |
B | LYS143 |
B | ALA144 |
B | GLY145 |
B | CYS147 |
B | HIS161 |
B | ILE162 |
B | GLY163 |
B | GLY164 |
B | ASN165 |
B | PHE170 |
B | EDO184 |
B | HOH314 |
B | HOH328 |
site_id | AC4 |
Number of Residues | 7 |
Details | BINDING SITE FOR RESIDUE EDO B 184 |
Chain | Residue |
B | GLN22 |
B | GLY23 |
B | HIS24 |
B | GLY145 |
B | HOH194 |
B | HOH259 |
B | AG7501 |