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3QOW

DOT1L Structure in complex with SAM

Functional Information from GO Data
ChainGOidnamespacecontents
A0031151molecular_functionhistone H3K79 methyltransferase activity
A0051726biological_processregulation of cell cycle
Functional Information from PDB Data
site_idAC1
Number of Residues21
DetailsBINDING SITE FOR RESIDUE SAM A 417
ChainResidue
APRO133
AVAL169
AGLU186
ALYS187
AGLY221
AASP222
APHE223
APHE239
AASN241
APHE245
AHOH441
AVAL135
AHOH464
AHOH524
AGLY137
AGLU138
ATHR139
AASP161
AGLY163
ASER164
AGLN168

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 418
ChainResidue
AARG203
AHIS213
AHOH448
AHOH553

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 419
ChainResidue
AARG229
AGLN252
AGLU255
AARG256

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues14
DetailsBinding site: {}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsModified residue: {"description":"Phosphoserine","evidences":[{"source":"PubMed","id":"23186163","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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