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3PK1

Crystal structure of Mcl-1 in complex with the BaxBH3 domain

Functional Information from GO Data
ChainGOidnamespacecontents
A0042981biological_processregulation of apoptotic process
B0042981biological_processregulation of apoptotic process
C0042981biological_processregulation of apoptotic process
D0042981biological_processregulation of apoptotic process
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CD A 1
ChainResidue
AGLU225
CHOH21
CHIS277
CHOH327

site_idAC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE CD A 2
ChainResidue
AHIS277
CHOH25
CGLU225

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CD A 5
ChainResidue
BGLU69
CASP304
AHOH23
AHIS224

site_idAC4
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CD A 12
ChainResidue
ACD14
ACYS286

site_idAC5
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CD A 13
ChainResidue
ACYS286
AGLU288

site_idAC6
Number of Residues3
DetailsBINDING SITE FOR RESIDUE CD A 14
ChainResidue
ACD12
AGLU240
ACYS286

site_idAC7
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CD A 17
ChainResidue
AGLU240
AASP241

site_idAC8
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CD A 18
ChainResidue
AGLU180
CGLU284

site_idAC9
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CD B 7
ChainResidue
BCD8
BCYS62

site_idBC1
Number of Residues3
DetailsBINDING SITE FOR RESIDUE CD B 8
ChainResidue
BCD7
BHOH18
BCYS62

site_idBC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CD C 3
ChainResidue
AASP304
CHOH22
CHIS224
DGLU69

site_idBC3
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CD C 4
ChainResidue
CHOH34
CHIS252

site_idBC4
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CD C 10
ChainResidue
CCD11
CCD15

site_idBC5
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CD C 11
ChainResidue
CCD10
CCYS286

site_idBC6
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CD C 15
ChainResidue
CCD10
CGLU240

site_idBC7
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CD C 16
ChainResidue
CGLU240
CASP241

site_idBC8
Number of Residues1
DetailsBINDING SITE FOR RESIDUE CD D 6
ChainResidue
DCYS62

site_idBC9
Number of Residues1
DetailsBINDING SITE FOR RESIDUE CD D 9
ChainResidue
DCYS62

Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues20
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. VFsDGvtNWGRIVTLIsFGA
ChainResidueDetails
AVAL253-ALA272

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WLvkqRGWDgFV
ChainResidueDetails
ATRP305-VAL316

site_idPS01259
Number of Residues15
DetailsBH3 Apoptosis regulator, Bcl-2 family BH3 motif signature. LsecLKrIGDELDSN
ChainResidueDetails
BLEU59-ASN73
AALA209-ASN223

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)
ChainResidueDetails
ALYS194
ALYS197
CLYS194
CLYS197

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PDB entries from 2024-07-24

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