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3PAG

Crystal structure of the V130D mutant of OXA-24/40 in complex with doripenem

Functional Information from GO Data
ChainGOidnamespacecontents
A0008658molecular_functionpenicillin binding
A0008800molecular_functionbeta-lactamase activity
A0016787molecular_functionhydrolase activity
A0071555biological_processcell wall organization
B0008658molecular_functionpenicillin binding
B0008800molecular_functionbeta-lactamase activity
B0016787molecular_functionhydrolase activity
B0071555biological_processcell wall organization
Functional Information from PDB Data
site_idAC1
Number of Residues13
DetailsBINDING SITE FOR RESIDUE 4J6 A 300
ChainResidue
AALA80
AGLY258
ASER259
AARG261
AHOH359
ASER81
ALEU127
ASER128
AASP130
ALEU168
ASER219
AGLY220
ATRP221

site_idAC2
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 1
ChainResidue
ALEU142
AGLU143
AHOH321

site_idAC3
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 2
ChainResidue
ALYS194
ALEU195
AHOH357

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 8
ChainResidue
AGLN178
AASN181
AHOH329
AHOH348
BGLN178

site_idAC5
Number of Residues13
DetailsBINDING SITE FOR RESIDUE 4J6 B 300
ChainResidue
BALA80
BSER81
BSER128
BASP130
BLEU168
BSER219
BGLY220
BTRP221
BGLY258
BSER259
BARG261
BHOH341
BHOH355

site_idAC6
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 B 4
ChainResidue
BGLY141
BLEU142
BGLU143
BHOH330

site_idAC7
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 B 5
ChainResidue
BTHR226
BPRO227
BGLN228
BHOH334
BHOH343

site_idAC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 B 7
ChainResidue
AGLN178
BGLN178
BASN181
BHOH277
BHOH328

225158

PDB entries from 2024-09-18

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