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3OZ1

cIAP1-BIR3 domain in complex with the Smac-mimetic compound Smac066

Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 501
ChainResidue
ACYS300
ACYS303
AHIS320
ACYS327

site_idAC2
Number of Residues10
DetailsBINDING SITE FOR RESIDUE BMB A 600
ChainResidue
AASP314
AGLU319
ATRP323
ALEU353
ALEU354
AGLY306
ALEU307
AARG308
ACYS309
AGLU311

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN B 501
ChainResidue
BCYS300
BCYS303
BHIS320
BCYS327

site_idAC4
Number of Residues8
DetailsBINDING SITE FOR RESIDUE BMB B 600
ChainResidue
BGLY306
BLEU307
BARG308
BCYS309
BGLU311
BASP314
BGLU319
BTRP323

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN C 501
ChainResidue
CCYS300
CCYS303
CHIS320
CCYS327

site_idAC6
Number of Residues8
DetailsBINDING SITE FOR RESIDUE BMB C 600
ChainResidue
CGLY306
CLEU307
CARG308
CCYS309
CGLU311
CASP314
CGLU319
CTRP323

site_idAC7
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN D 501
ChainResidue
DCYS300
DCYS303
DHIS320
DCYS327

site_idAC8
Number of Residues9
DetailsBINDING SITE FOR RESIDUE BMB D 600
ChainResidue
DGLY306
DLEU307
DARG308
DCYS309
DTRP310
DASP314
DGLU319
DTRP323
DLEU353

Functional Information from PROSITE/UniProt
site_idPS01282
Number of Residues68
DetailsBIR_REPEAT_1 BIR repeat. HaaRmrtfmy.Wpssvpvqpeqlas.AGFyYvgrnDdvkCfcCdgglrcWesgddpwveHakwfPrCefL
ChainResidueDetails
AHIS263-LEU330

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues16
DetailsBINDING:
ChainResidueDetails
ACYS300
CCYS303
CHIS320
CCYS327
DCYS300
DCYS303
DHIS320
DCYS327
ACYS303
AHIS320
ACYS327
BCYS300
BCYS303
BHIS320
BCYS327
CCYS300

221716

PDB entries from 2024-06-26

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