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3OMO

Fragment-Based Design of novel Estrogen Receptor Ligands

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues11
DetailsBINDING SITE FOR RESIDUE WV7 A 1
ChainResidue
ALEU298
ALEU476
AHOH504
AGLU305
ALEU339
AMET340
AARG346
APHE356
AILE373
AILE376
AGLY472

site_idAC2
Number of Residues10
DetailsBINDING SITE FOR RESIDUE WV7 B 1
ChainResidue
BHOH73
BLEU298
BGLU305
BLEU339
BARG346
BPHE356
BILE373
BILE376
BGLY472
BLEU476

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
CSER13
DSER13

221051

PDB entries from 2024-06-12

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