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3OMJ

Structural Basis for Cyclic Py-Im Polyamide Allosteric Inhibition of Nuclear Receptor Binding

Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE CA A 302
ChainResidue
AHOH124
AHOH246
AHOH247
AHOH252
AHOH253
BHOH125
BHOH245

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CA A 300
ChainResidue
AHOH73
AHOH74
AHOH133
AHOH161
AHOH32
AHOH34

site_idAC3
Number of Residues7
DetailsBINDING SITE FOR RESIDUE CA A 301
ChainResidue
AHOH32
AHOH34
AHOH41
AHOH73
AHOH74
AHOH133
AHOH161

site_idAC4
Number of Residues39
DetailsBINDING SITE FOR RESIDUE 1P2 B 500
ChainResidue
ADC1
ADG4
ADT5
ADA6
ADC7
ADT8
ADG9
AHOH160
AHOH242
BDC1
BDG4
BDT5
BDA6
BDC7
BDT8
BDG9
BDG10
BHOH31
BHOH39
BHOH40
BHOH47
BHOH53
BHOH56
BHOH86
BHOH87
BHOH102
BHOH129
BHOH137
BHOH138
BHOH146
BHOH159
BHOH169
BHOH170
BHOH176
BHOH182
BHOH198
BHOH200
BHOH203
BHOH204

site_idAC5
Number of Residues6
DetailsBINDING SITE FOR RESIDUE CA B 303
ChainResidue
BC382
BC382
BHOH45
BHOH45
BHOH85
BHOH85

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PDB entries from 2024-05-01

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