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3NJQ

Crystal structure of Kaposi's sarcoma-associated herpesvirus protease in complex with dimer disruptor

Functional Information from GO Data
ChainGOidnamespacecontents
A0004252molecular_functionserine-type endopeptidase activity
A0006508biological_processproteolysis
B0004252molecular_functionserine-type endopeptidase activity
B0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE ACT A 1
ChainResidue
AGLU100
ALEU103
AGLY151
AHIS152
ATRP156

site_idAC2
Number of Residues13
DetailsBINDING SITE FOR RESIDUE NJQ A 197
ChainResidue
APHE189
APRO192
AHOH219
BLEU47
BTHR195
BLEU196
BNJQ198
BNJQ199
BHOH206
APHE76
ALEU79
AILE105
ATRP109

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 B 1
ChainResidue
BHIS88
BARG91
BARG91
BHOH254

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 B 2
ChainResidue
AVAL89
AALA92
BTHR108
BTRP109
BARG143

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 B 3
ChainResidue
ALYS99
AHOH229
BTRP156
BARG160

site_idAC6
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL B 197
ChainResidue
AGLN133
AHOH223
BLEU184
BSER185
BHOH256

site_idAC7
Number of Residues16
DetailsBINDING SITE FOR RESIDUE NJQ B 198
ChainResidue
ALYS18
ATRP109
AALA139
ANJQ197
BLEU79
BLEU83
BVAL89
BALA90
BILE105
BLEU106
BTRP109
BSER191
BPRO192
BLEU193
BNJQ199
BHOH252

site_idAC8
Number of Residues13
DetailsBINDING SITE FOR RESIDUE NJQ B 199
ChainResidue
ALEU83
ASER87
AVAL89
ATRP109
ALEU193
ANJQ197
BGLU45
BLEU47
BLEU140
BARG144
BNJQ198
BHOH228
BHOH244

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PDB entries from 2024-07-24

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