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3MF5

Hepatitis C virus polymerase NS5B (BK) with amide bioisostere thumb site inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003723molecular_functionRNA binding
A0003968molecular_functionRNA-dependent RNA polymerase activity
A0039694biological_processviral RNA genome replication
B0003723molecular_functionRNA binding
B0003968molecular_functionRNA-dependent RNA polymerase activity
B0039694biological_processviral RNA genome replication
Functional Information from PDB Data
site_idAC1
Number of Residues9
DetailsBINDING SITE FOR RESIDUE HJZ A 571
ChainResidue
AARG422
AMET423
ASER476
ATYR477
AILE482
ALEU497
AARG501
ATRP528
AHOH788

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL A 602
ChainResidue
AGLU143
AVAL144
AARG394
AGLU398
AHOH642

site_idAC3
Number of Residues8
DetailsBINDING SITE FOR RESIDUE HJZ B 571
ChainResidue
BLEU419
BARG422
BSER476
BTYR477
BILE482
BARG501
BTRP528
BHOH713

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000305|PubMed:10557268, ECO:0000305|PubMed:11884572
ChainResidueDetails
AASP220
AASP318
AASP319
BASP220
BASP318
BASP319

site_idSWS_FT_FI2
Number of Residues4
DetailsMOD_RES: Phosphoserine; by host => ECO:0000250|UniProtKB:P26662
ChainResidueDetails
ASER29
ASER42
BSER29
BSER42

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PDB entries from 2024-06-12

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