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3L0E

X-ray crystal structure of a Potent Liver X Receptor Modulator

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006629biological_processlipid metabolic process
Functional Information from PDB Data
site_idAC1
Number of Residues20
DetailsBINDING SITE FOR RESIDUE G58 A 1
ChainResidue
APHE268
AARG319
APHE329
ALEU330
APHE340
AALA343
AGLY344
ALEU345
AHIS435
ALEU442
ALEU453
APHE271
ATRP457
ATHR272
ALEU274
AALA275
ASER278
AILE309
AMET312
ATHR316

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues238
DetailsDomain: {"description":"NR LBD","evidences":[{"source":"PROSITE-ProRule","id":"PRU01189","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues241
DetailsRegion: {"description":"Transactivation AF-2; required for ligand-dependent transactivation function; mediates interaction with CCAR2","evidences":[{"source":"PubMed","id":"25661920","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues3
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2)","evidences":[{"source":"PubMed","id":"20159957","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 3"}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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