3L03
Crystal Structure of human Estrogen Receptor alpha Ligand-Binding Domain in complex with a Glucocorticoid Receptor Interacting Protein 1 Nr Box II peptide and Estetrol (Estra-1,3,5(10)-triene-3,15 alpha,16alpha,17beta-tetrol)
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 4 |
Details | BINDING SITE FOR RESIDUE CL A 1 |
Chain | Residue |
A | HOH18 |
A | HOH54 |
A | ARG352 |
B | ARG352 |
site_id | AC2 |
Number of Residues | 5 |
Details | BINDING SITE FOR RESIDUE GOL A 2 |
Chain | Residue |
A | ASN439 |
A | GLN441 |
A | GLU444 |
A | ALA493 |
A | LEU495 |
site_id | AC3 |
Number of Residues | 12 |
Details | BINDING SITE FOR RESIDUE 4OH A 551 |
Chain | Residue |
A | HOH3 |
A | MET343 |
A | LEU346 |
A | GLU353 |
A | LEU387 |
A | MET388 |
A | ARG394 |
A | PHE404 |
A | ILE424 |
A | GLY521 |
A | HIS524 |
A | LEU525 |
site_id | AC4 |
Number of Residues | 10 |
Details | BINDING SITE FOR RESIDUE 4OH B 2 |
Chain | Residue |
B | HOH23 |
B | MET343 |
B | LEU346 |
B | GLU353 |
B | LEU387 |
B | ARG394 |
B | ILE424 |
B | GLY521 |
B | HIS524 |
B | LEU525 |
Functional Information from SwissProt/UniProt
Chain | Residue | Details |
A | SER537 | |
B | SER537 | |
site_id | SWS_FT_FI2 |
Number of Residues | 2 |
Details | LIPID: S-palmitoyl cysteine => ECO:0000250 |
Chain | Residue | Details |
A | CYS447 | |
B | CYS447 | |