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3IA9

Crystal structure of a chemically synthesized [D25N]HIV-1 protease molecule complexed with MVT-101 reduced isostere inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0004190molecular_functionaspartic-type endopeptidase activity
A0006508biological_processproteolysis
B0004190molecular_functionaspartic-type endopeptidase activity
B0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues35
DetailsBINDING SITE FOR RESIDUE 2NC A 100
ChainResidue
AASN25
APHE53
AVAL82
AILE84
AHOH101
AHOH107
AHOH109
AHOH112
AHOH118
AHOH128
AHOH139
AGLY27
AHOH148
BLEU23
BASN25
BGLY27
BALA28
BASP29
BASP30
BNLE46
BILE47
BGLY48
AALA28
BGLY49
BILE50
BPHE53
BPRO81
BILE84
BHOH121
AASP29
AASP30
AILE47
AGLY48
AGLY49
AILE50

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 401
ChainResidue
ALEU10
AGLU21
AALA22
AVAL82
AASN83
AHOH106

site_idAC3
Number of Residues10
DetailsBINDING SITE FOR RESIDUE SO4 A 402
ChainResidue
ATHR12
AILE13
AARG14
ALEU19
ATRP42
APRO44
AGLU65
AILE66
AABA67
AGLY68

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PDB entries from 2024-10-09

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