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3HZF

Structure of TR-alfa bound to selective thyromimetic GC-1 in C2 space group

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues12
DetailsBINDING SITE FOR RESIDUE B72 A 1
ChainResidue
AILE222
ALEU292
AHIS381
APHE401
AALA225
AARG228
AMET256
AMET259
ALEU276
ASER277
AGLY290
AGLY291

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsBINDING: BINDING => ECO:0000269|PubMed:16781732, ECO:0007744|PDB:2H77, ECO:0007744|PDB:2H79
ChainResidueDetails
AARG228

site_idSWS_FT_FI2
Number of Residues1
DetailsBINDING: BINDING => ECO:0000269|PubMed:16781732, ECO:0007744|PDB:2H79
ChainResidueDetails
ASER277

223790

PDB entries from 2024-08-14

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