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3HVL

Tethered PXR-LBD/SRC-1p complexed with SR-12813

Replaces:  3CTC
Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues16
DetailsBINDING SITE FOR RESIDUE SRL A 1
ChainResidue
AHOH93
ATYR306
AMET323
AHIS407
ALEU411
APHE420
AMET425
APHE429
AMET243
AMET246
ASER247
APHE251
APHE281
AGLN285
APHE288
ATRP299

site_idAC2
Number of Residues15
DetailsBINDING SITE FOR RESIDUE SRL B 2
ChainResidue
BALA244
BSER247
BPHE251
BPHE281
BGLN285
BTRP299
BTYR306
BMET323
BHIS327
BHIS407
BLEU411
BPHE420
BPHE429
BHOH471
BHOH503

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
ChainResidueDetails
ASER247
AGLN285
AHIS407
BSER247
BGLN285
BHIS407

site_idSWS_FT_FI2
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ASER460
BSER460

218853

PDB entries from 2024-04-24

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