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3HVL

Tethered PXR-LBD/SRC-1p complexed with SR-12813

Replaces:  3CTC
Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues16
DetailsBINDING SITE FOR RESIDUE SRL A 1
ChainResidue
AHOH93
ATYR306
AMET323
AHIS407
ALEU411
APHE420
AMET425
APHE429
AMET243
AMET246
ASER247
APHE251
APHE281
AGLN285
APHE288
ATRP299

site_idAC2
Number of Residues15
DetailsBINDING SITE FOR RESIDUE SRL B 2
ChainResidue
BALA244
BSER247
BPHE251
BPHE281
BGLN285
BTRP299
BTYR306
BMET323
BHIS327
BHIS407
BLEU411
BPHE420
BPHE429
BHOH471
BHOH503

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues10
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"12578355","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1M13","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues8
DetailsMotif: {"description":"LXXLL motif 4"}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues1
DetailsModified residue: {"description":"Phosphoserine","evidences":[{"source":"PubMed","id":"23186163","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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