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3H82

Crystal structure of the high affinity heterodimer of HIF2 alpha and ARNT C-terminal PAS domains with the artificial ligand THS020

Functional Information from PDB Data
site_idAC1
Number of Residues15
DetailsBINDING SITE FOR RESIDUE 020 A 351
ChainResidue
AHIS248
ATYR307
AMET309
ATHR321
AILE337
ACYS339
AASN341
AMET252
APHE254
AALA277
ATYR281
AMET289
ASER292
AVAL302
ASER304

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues86
DetailsDomain: {"description":"PAC"}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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