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3GGX

HIV Protease, pseudo-symmetric inhibitors

Functional Information from GO Data
ChainGOidnamespacecontents
A0004190molecular_functionaspartic-type endopeptidase activity
A0006508biological_processproteolysis
B0004190molecular_functionaspartic-type endopeptidase activity
B0006508biological_processproteolysis
C0004190molecular_functionaspartic-type endopeptidase activity
C0006508biological_processproteolysis
D0004190molecular_functionaspartic-type endopeptidase activity
D0006508biological_processproteolysis
E0004190molecular_functionaspartic-type endopeptidase activity
E0006508biological_processproteolysis
F0004190molecular_functionaspartic-type endopeptidase activity
F0006508biological_processproteolysis
G0004190molecular_functionaspartic-type endopeptidase activity
G0006508biological_processproteolysis
H0004190molecular_functionaspartic-type endopeptidase activity
H0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues16
DetailsBINDING SITE FOR RESIDUE GGX H 1001
ChainResidue
GARG8
HASP25
HGLY27
HALA28
HASP29
HGLY48
HGLY49
HVAL82
GLEU23
GASP25
GGLY27
GASP29
GGLY48
GGLY49
GPRO81
HARG8

site_idAC2
Number of Residues17
DetailsBINDING SITE FOR RESIDUE GGX B 1002
ChainResidue
AARG8
ALEU23
AASP25
AGLY27
AALA28
AASP29
AGLY48
AGLY49
APRO81
BARG8
BLEU23
BASP25
BGLY27
BASP29
BGLY48
BGLY49
BILE50

site_idAC3
Number of Residues19
DetailsBINDING SITE FOR RESIDUE GGX E 1003
ChainResidue
EARG8
EASP25
EGLY27
EALA28
EASP29
EGLY48
EGLY49
EILE50
EVAL82
FARG8
FASP25
FGLY27
FALA28
FASP29
FGLY48
FGLY49
FILE50
FPRO81
FILE84

site_idAC4
Number of Residues16
DetailsBINDING SITE FOR RESIDUE GGX C 1004
ChainResidue
CARG8
CASP25
CGLY27
CALA28
CASP29
CGLY48
CGLY49
CILE84
DARG8
DLEU23
DASP25
DGLY27
DALA28
DASP29
DGLY48
DGLY49

Functional Information from PROSITE/UniProt
site_idPS00141
Number of Residues12
DetailsASP_PROTEASE Eukaryotic and viral aspartyl proteases active site. ALLDTGADDTVL
ChainResidueDetails
AALA22-LEU33

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsACT_SITE: For protease activity; shared with dimeric partner => ECO:0000255|PROSITE-ProRule:PRU10094, ECO:0000269|PubMed:12924029
ChainResidueDetails
AASP25
BASP25
CASP25
DASP25
EASP25
FASP25
GASP25
HASP25

site_idSWS_FT_FI2
Number of Residues8
DetailsSITE: Cleavage; by viral protease => ECO:0000269|PubMed:2476069
ChainResidueDetails
APHE99
BPHE99
CPHE99
DPHE99
EPHE99
FPHE99
GPHE99
HPHE99

Catalytic Information from CSA
site_idCSA1
Number of Residues2
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
AASP25
ATHR26

site_idCSA10
Number of Residues1
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
BASP25

site_idCSA11
Number of Residues1
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
CASP25

site_idCSA12
Number of Residues1
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
DASP25

site_idCSA13
Number of Residues1
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
EASP25

site_idCSA14
Number of Residues1
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
FASP25

site_idCSA15
Number of Residues1
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
GASP25

site_idCSA16
Number of Residues1
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
HASP25

site_idCSA2
Number of Residues2
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
BASP25
BTHR26

site_idCSA3
Number of Residues2
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
CASP25
CTHR26

site_idCSA4
Number of Residues2
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
DASP25
DTHR26

site_idCSA5
Number of Residues2
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
EASP25
ETHR26

site_idCSA6
Number of Residues2
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
FASP25
FTHR26

site_idCSA7
Number of Residues2
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
GASP25
GTHR26

site_idCSA8
Number of Residues2
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
HASP25
HTHR26

site_idCSA9
Number of Residues1
DetailsAnnotated By Reference To The Literature 1a30
ChainResidueDetails
AASP25

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PDB entries from 2024-09-11

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