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3FSI

Crystal structure of a trypanocidal 4,4'-Bis(imidazolinylamino)diphenylamine bound to DNA

Functional Information from PDB Data
site_idAC1
Number of Residues2
DetailsBINDING SITE FOR RESIDUE ACT A 378
ChainResidue
AGLN91
ASER92

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE ACT A 379
ChainResidue
AASP153
AALA154
APHE155
APHE156
AGLN190
AHOH303

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE ACT A 380
ChainResidue
APRO127
ATHR197
AHOH283
AHOH431
AILE125

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ACT A 381
ChainResidue
AMET66
AGLU171
ATRP172
AARG173

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ACT A 382
ChainResidue
ATHR24
ATRP25
APHE29
AARG241

site_idAC6
Number of Residues10
DetailsBINDING SITE FOR RESIDUE MWB G 9
ChainResidue
BDA10
BDA11
BDT12
BDT13
BDA14
GDA4
GDA5
GDT6
GDT7
GDC8

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Cleavage; by viral protease => ECO:0000269|PubMed:16603535
ChainResidueDetails
AASN95

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphoserine; by host => ECO:0000305|PubMed:12525616
ChainResidueDetails
ALEU72

218196

PDB entries from 2024-04-10

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