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3FNU

Crystal structure of KNI-10006 bound histo-aspartic protease (HAP) from Plasmodium falciparum

Functional Information from GO Data
ChainGOidnamespacecontents
A0004190molecular_functionaspartic-type endopeptidase activity
A0006508biological_processproteolysis
B0004190molecular_functionaspartic-type endopeptidase activity
B0006508biological_processproteolysis
C0004190molecular_functionaspartic-type endopeptidase activity
C0006508biological_processproteolysis
D0004190molecular_functionaspartic-type endopeptidase activity
D0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues9
DetailsBINDING SITE FOR RESIDUE 006 A 329
ChainResidue
AALA10
AVAL12
APHE109
APHE111
ATYR112
AVAL120
AALA217
AHOH349
AHOH351

site_idAC2
Number of Residues9
DetailsBINDING SITE FOR RESIDUE 006 B 329
ChainResidue
BALA10
BVAL12
BTRP39
BILE80
BPHE109
BPHE111
BVAL120
BALA217
BHOH359

site_idAC3
Number of Residues7
DetailsBINDING SITE FOR RESIDUE 006 C 329
ChainResidue
CVAL12
CSER35
CTRP39
CLEU73
CPHE109
CPHE111
CALA217

site_idAC4
Number of Residues11
DetailsBINDING SITE FOR RESIDUE 006 D 329
ChainResidue
DVAL12
DSER35
DTRP39
DLEU73
DILE80
DMET104
DILE107
DPHE109
DPHE111
DTYR112
DALA217

Catalytic Information from CSA
site_idCSA1
Number of Residues4
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
AASP215
ASER35
ATHR218
AHIS32

site_idCSA10
Number of Residues4
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
BASP215
BTHR218
BHIS32
BTHR33

site_idCSA11
Number of Residues4
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
CASP215
CTHR218
CHIS32
CTHR33

site_idCSA12
Number of Residues4
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
DASP215
DTHR218
DHIS32
DTHR33

site_idCSA13
Number of Residues1
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
AHIS32

site_idCSA14
Number of Residues1
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
BHIS32

site_idCSA15
Number of Residues1
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
CHIS32

site_idCSA16
Number of Residues1
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
DHIS32

site_idCSA17
Number of Residues1
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
AASP215

site_idCSA18
Number of Residues1
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
BASP215

site_idCSA19
Number of Residues1
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
CASP215

site_idCSA2
Number of Residues4
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
BASP215
BSER35
BTHR218
BHIS32

site_idCSA20
Number of Residues1
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
DASP215

site_idCSA3
Number of Residues4
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
CASP215
CSER35
CTHR218
CHIS32

site_idCSA4
Number of Residues4
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
DASP215
DSER35
DTHR218
DHIS32

site_idCSA5
Number of Residues3
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
AASP215
ASER35
AHIS32

site_idCSA6
Number of Residues3
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
BASP215
BSER35
BHIS32

site_idCSA7
Number of Residues3
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
CASP215
CSER35
CHIS32

site_idCSA8
Number of Residues3
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
DASP215
DSER35
DHIS32

site_idCSA9
Number of Residues4
DetailsAnnotated By Reference To The Literature 1am5
ChainResidueDetails
AASP215
ATHR218
AHIS32
ATHR33

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PDB entries from 2024-07-10

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