Loading
PDBj
MenuPDBj@FacebookPDBj@X(formerly Twitter)PDBj@BlueSkyPDBj@YouTubewwPDB FoundationwwPDBDonate
RCSB PDBPDBeBMRBAdv. SearchSearch help

3ET2

Structure of PPARdelta with 3-[5-Methoxy-1-(4-methoxy-benzenesulfonyl)-1H-indol-3-yl]-propionic acid

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues14
DetailsBINDING SITE FOR RESIDUE ET1 A 1
ChainResidue
APHE246
AMET417
ALEU433
ATYR437
AHOH444
AHOH534
ACYS249
ATHR253
AHIS287
APHE291
APHE324
AILE327
ALYS331
AHIS413

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE 1BO A 3
ChainResidue
ATHR261
ALEU282
BPHE274
BLEU275

site_idAC3
Number of Residues2
DetailsBINDING SITE FOR RESIDUE 1BO A 4
ChainResidue
ALEU275
BTHR261

site_idAC4
Number of Residues3
DetailsBINDING SITE FOR RESIDUE 1BO A 6
ChainResidue
ALEU219
ATRP220
AILE241

site_idAC5
Number of Residues19
DetailsBINDING SITE FOR RESIDUE ET1 B 2
ChainResidue
BPHE246
BCYS249
BGLN250
BTHR252
BTHR253
BHIS287
BILE290
BPHE291
BLEU294
BPHE324
BILE327
BILE328
BLYS331
BHIS413
BMET417
BLEU433
BTYR437
BHOH461
BHOH576

238268

PDB entries from 2025-07-02

PDB statisticsPDBj update infoContact PDBjnumon