Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

3ECN

Crystal structure of PDE8A catalytic domain in complex with IBMX

Functional Information from GO Data
ChainGOidnamespacecontents
A0004114molecular_function3',5'-cyclic-nucleotide phosphodiesterase activity
A0007165biological_processsignal transduction
A0008081molecular_functionphosphoric diester hydrolase activity
B0004114molecular_function3',5'-cyclic-nucleotide phosphodiesterase activity
B0007165biological_processsignal transduction
B0008081molecular_functionphosphoric diester hydrolase activity
Functional Information from PDB Data
site_idAC1
Number of Residues8
DetailsBINDING SITE FOR RESIDUE IBM A 3
ChainResidue
AMET670
AILE744
ATYR748
APHE767
AGLN778
APHE781
APHE785
AHOH884

site_idAC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE IBM B 3
ChainResidue
BMET670
BILE744
BTYR748
BGLN778
BPHE781
BPHE785
BHOH126

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE ZN A 1
ChainResidue
AHIS560
AHIS596
AASP597
AASP726
AHOH820
AHOH821

site_idAC4
Number of Residues6
DetailsBINDING SITE FOR RESIDUE MG A 2
ChainResidue
AASP597
AHOH820
AHOH822
AHOH823
AHOH824
AHOH825

site_idAC5
Number of Residues6
DetailsBINDING SITE FOR RESIDUE ZN B 1
ChainResidue
BHOH11
BHOH12
BHIS560
BHIS596
BASP597
BASP726

site_idAC6
Number of Residues6
DetailsBINDING SITE FOR RESIDUE MG B 2
ChainResidue
BHOH11
BHOH13
BHOH14
BHOH15
BHOH16
BASP597

Functional Information from PROSITE/UniProt
site_idPS00126
Number of Residues12
DetailsPDEASE_I_1 3'5'-cyclic nucleotide phosphodiesterase domain signature. HDVdHpGrtNsF
ChainResidueDetails
AHIS596-PHE607

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsACT_SITE: Proton donor => ECO:0000250|UniProtKB:O76083
ChainResidueDetails
AHIS556
BHIS556

site_idSWS_FT_FI2
Number of Residues8
DetailsBINDING: BINDING => ECO:0000269|PubMed:18983167, ECO:0007744|PDB:3ECM, ECO:0007744|PDB:3ECN
ChainResidueDetails
AHIS560
AHIS596
AASP597
AASP726
BHIS560
BHIS596
BASP597
BASP726

219140

PDB entries from 2024-05-01

PDB statisticsPDBj update infoContact PDBjnumon