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3CWJ

Crystal structure of hcv ns5b polymerase with a novel pyridazinone inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003723molecular_functionRNA binding
A0003968molecular_functionRNA-dependent RNA polymerase activity
A0039694biological_processviral RNA genome replication
B0003723molecular_functionRNA binding
B0003968molecular_functionRNA-dependent RNA polymerase activity
B0039694biological_processviral RNA genome replication
Functional Information from PDB Data
site_idAC1
Number of Residues16
DetailsBINDING SITE FOR RESIDUE 321 A 1001
ChainResidue
APHE193
AASN411
AMET414
ATYR415
AGLN446
ATYR448
ASER556
AHOH1096
ASER288
AASN291
AASN316
AASP318
ACYS366
ASER368
ALEU384
AGLY410

site_idAC2
Number of Residues20
DetailsBINDING SITE FOR RESIDUE 321 B 1002
ChainResidue
BPHE193
BARG200
BSER288
BASN291
BASN316
BGLY317
BASP318
BCYS366
BSER368
BLEU384
BGLY410
BASN411
BMET414
BTYR415
BGLN446
BTYR448
BGLY449
BSER556
BHOH1036
BHOH1081

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000305|PubMed:10557268, ECO:0000305|PubMed:11884572
ChainResidueDetails
AASP220
AASP318
AASP319
BASP220
BASP318
BASP319

site_idSWS_FT_FI2
Number of Residues4
DetailsMOD_RES: Phosphoserine; by host => ECO:0000250|UniProtKB:P26662
ChainResidueDetails
ASER29
ASER42
BSER29
BSER42

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PDB entries from 2024-07-10

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