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3BSC

Crystal Structure of HCV NS5B Polymerase with a Novel Pyridazinone Inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003723molecular_functionRNA binding
A0003968molecular_functionRNA-dependent RNA polymerase activity
A0039694biological_processviral RNA genome replication
B0003723molecular_functionRNA binding
B0003968molecular_functionRNA-dependent RNA polymerase activity
B0039694biological_processviral RNA genome replication
Functional Information from PDB Data
site_idAC1
Number of Residues19
DetailsBINDING SITE FOR RESIDUE 2PD A 579
ChainResidue
APHE193
AGLY410
AASN411
AMET414
ATYR415
AGLN446
ATYR448
AGLY449
ASER556
AHOH662
AHOH666
APRO197
AARG200
AASN316
AGLY317
AASP318
ACYS366
ASER368
ALEU384

site_idAC2
Number of Residues17
DetailsBINDING SITE FOR RESIDUE 2PD B 579
ChainResidue
BPHE193
BPRO197
BARG200
BASN316
BASP318
BCYS366
BSER368
BLEU384
BGLY410
BASN411
BTYR415
BGLN446
BTYR448
BGLY449
BSER556
BHOH641
BHOH658

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000305|PubMed:10557268, ECO:0000305|PubMed:11884572
ChainResidueDetails
AASP220
AASP318
AASP319
BASP220
BASP318
BASP319

site_idSWS_FT_FI2
Number of Residues4
DetailsMOD_RES: Phosphoserine; by host => ECO:0000250|UniProtKB:P26662
ChainResidueDetails
ASER29
ASER42
BSER29
BSER42

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PDB entries from 2024-09-11

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