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3ADS

Human PPARgamma ligand-binding domain in complex with indomethacin

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues10
DetailsBINDING SITE FOR RESIDUE IMN A 1
ChainResidue
AARG280
AMET364
AGLY284
ACYS285
AARG288
ALEU330
ALEU340
AILE341
ASER342
AMET348

site_idAC2
Number of Residues15
DetailsBINDING SITE FOR RESIDUE IMN A 2
ChainResidue
AILE281
APHE282
ACYS285
ASER289
AHIS323
ATYR327
ALEU330
ALEU356
APHE360
APHE363
AMET364
AHIS449
ALEU453
ALEU469
ATYR473

site_idAC3
Number of Residues11
DetailsBINDING SITE FOR RESIDUE IMN B 3
ChainResidue
BILE281
BARG288
BSER289
BALA292
BILE326
BLEU330
BLEU333
BLEU340
BILE341
BGLU343
BMET364

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsMotif: {"description":"9aaTAD","evidences":[{"source":"PubMed","id":"30468856","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues12
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"9744270","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"2PRG","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues4
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)","evidences":[{"source":"PubMed","id":"36737649","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

243083

PDB entries from 2025-10-15

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