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3A78

Crystal structure of the human VDR ligand binding domain bound to the natural metabolite 1alpha,25-dihydroxy-3-epi-vitamin D3

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues14
DetailsBINDING SITE FOR RESIDUE 3EV A 428
ChainResidue
AHOH9
ASER278
ATRP286
ACYS288
AHIS305
AHIS397
ATYR143
ATYR147
ALEU227
AVAL234
ASER237
AILE271
AARG274
ASER275

site_idAC2
Number of Residues8
DetailsBINDING SITE FOR RESIDUE SO4 A 1
ChainResidue
AHOH56
AHOH184
APRO408
AGLU409
ACYS410
ASER411
AHOH458
AHOH498

site_idAC3
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 2
ChainResidue
ATHR280
AMET281
ALYS321

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsBINDING: BINDING => ECO:0000269|PubMed:10678179, ECO:0000269|PubMed:11344298
ChainResidueDetails
ATYR143
ALEU227
AILE271
AHIS305
AHIS397

219140

PDB entries from 2024-05-01

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