3A3Z
Crystal structure of the human VDR ligand binding domain bound to the synthetic agonist compound 2alpha-methyl-AMCR277A(C23S)
Functional Information from GO Data
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 11 |
Details | BINDING SITE FOR RESIDUE 2MV X 1 |
Chain | Residue |
X | TYR143 |
X | HIS305 |
X | HIS397 |
X | LEU227 |
X | VAL234 |
X | SER237 |
X | ARG274 |
X | SER275 |
X | SER278 |
X | TRP286 |
X | CYS288 |
site_id | AC2 |
Number of Residues | 10 |
Details | BINDING SITE FOR RESIDUE SO4 X 428 |
Chain | Residue |
X | HOH32 |
X | HOH200 |
X | PRO408 |
X | GLU409 |
X | CYS410 |
X | SER411 |
X | MET412 |
X | HOH498 |
X | HOH584 |
X | HOH683 |
site_id | AC3 |
Number of Residues | 4 |
Details | BINDING SITE FOR RESIDUE SO4 X 2 |
Chain | Residue |
X | THR280 |
X | MET281 |
X | LYS321 |
X | HOH438 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 2 |
Details | BINDING: BINDING => ECO:0000269|PubMed:10678179, ECO:0000269|PubMed:11344298, ECO:0007744|PDB:1DB1, ECO:0007744|PDB:1IE8 |
Chain | Residue | Details |
X | TYR143 | |
X | LEU325 |
site_id | SWS_FT_FI2 |
Number of Residues | 1 |
Details | BINDING: BINDING => ECO:0000269|PubMed:10678179, ECO:0000269|PubMed:11344298, ECO:0007744|PDB:1DB1 |
Chain | Residue | Details |
X | CYS288 |
site_id | SWS_FT_FI3 |
Number of Residues | 2 |
Details | BINDING: BINDING => ECO:0000269|PubMed:10678179, ECO:0000269|PubMed:11344298, ECO:0007744|PDB:1IE8 |
Chain | Residue | Details |
X | GLU329 | |
X | GLN356 |
site_id | SWS_FT_FI4 |
Number of Residues | 1 |
Details | BINDING: BINDING => ECO:0000269|PubMed:10678179, ECO:0000269|PubMed:11344298 |
Chain | Residue | Details |