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2REW

Crystal Structure of PPARalpha ligand binding domain with BMS-631707

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues8
DetailsBINDING SITE FOR RESIDUE CPQ A 1
ChainResidue
ALYS204
AALA207
ALYS208
AARG348
ASER373
ALEU410
AHIS411
AGLU451

site_idAC2
Number of Residues15
DetailsBINDING SITE FOR RESIDUE REW A 469
ChainResidue
ACYS275
ACYS276
AGLN277
ASER280
ATYR314
AMET330
AVAL332
AILE354
AHIS440
AILE447
ALEU456
ALEU460
ATYR464
AHOH527
APHE273

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:19116277, ECO:0007744|PDB:3ET1
ChainResidueDetails
ASER280
ATYR314
ATYR464

site_idSWS_FT_FI2
Number of Residues1
DetailsSITE: Essential for heterodimerization with RXRA
ChainResidueDetails
ALEU433

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PDB entries from 2024-07-17

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